Radical Reactions and Bond Cleavage

Jul 15, 2024

Radical Reactions and Bond Cleavage

Introduction

  • Topic: Radical reactions
  • Key Concepts: Bonds breaking, homolytic and heterolytic cleavage, geometric implications, stability, and resonance.

Bond Cleavage

Heterolytic Cleavage

  • Induced by: Heat (Delta symbol)
  • Process: Both electrons in a bond move to one atom, forming ionic species ( + and - charges).
  • Representation: Double barbed arrow.

Homolytic Cleavage

  • Induced by: Light
  • Process: Electrons in a bond split, one electron going to each atom forming radicals.
  • Representation: Single barbed arrows leading to neutral species with unpaired electrons.

Radical Geometry

  • Carbocation Geometry (SP2)
    • Example: Tertiary carbocation (three methyl groups in the same plane)
    • Hybridization: SP2
    • Empty P Orbital: Perpendicular to the plane
  • Anion Geometry (SP3)
    • P Orbital filled with lone pairs
    • Shape: Trigonal pyramidal due to lone pairs repelling bond pairs

Radical Characteristics

  • Radical Species: Neutral with one unpaired electron
  • Geometry: Between planar (sp2) and trigonal pyramidal (sp3), but often assumed to be planar.
  • Radical Stability: Follows similar order as carbocations due to hyperconjugation.

Stability Trends

  • Methyl radical < Primary radical < Secondary radical < Tertiary radical due to hyperconjugation.

Bond Dissociation Energies

  • Significance: Energy required to break a bond homolytically
  • Example:
    • Methane: 435 kJ/mol
    • Tertiary radical: 381 kJ/mol
  • Trends: Lower energy indicates more stable radicals

Resonance Structures in Radicals

  • Allylic Radicals: Stabilized by resonance
  • Benzylic Radicals: Extremely stabilized by resonance compared to allylic

Special Case: Vinylic Radicals

  • Energy: 464 kJ/mol, thus very unstable

Radical Reactions

No Rearrangements

  • Unlike carbocations, radicals don't typically rearrange.

Patterns of Radical Reactions

1. Homolytic Bond Cleavage

  • Example: X-Y bond cleavage under light or heat to form radicals.

2. Addition to a Pi Bond

  • Example: Radical adds to a double bond, forming a new radical on the adjacent carbon.

3. Hydrogen Abstraction

  • Example: Radical abstracts a hydrogen from another molecule, forming a new radical.

4. Halogen Abstraction

  • Example: Alkyl radical abstracts a halogen atom from a molecule.

5. Elimination

  • Example: Radical removes itself as a pi bond forms on the adjacent carbons.

6. Coupling

  • Example: Two radicals combine to form a covalent bond.

Stages of Radical Reactions

Initiation

  • Description: Formation of radical species to start the reaction.
  • Example: Homolytic cleavage.

Propagation

  • Description: Radicals react with molecules to form new radicals and continue the reaction.
  • Utilizes: Hydrogen and halogen abstraction, addition to a pi bond, and elimination.

Termination

  • Description: Radicals combine and neutralize each other to end the reaction.
  • Example: Coupling.

Summary

  • Radical reactions are critical in chemistry, involving specific steps and patterns. Understanding bond dissociation energies, geometry, and stability trends is essential for mastering the behavior of radicals in various reactions.