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Neurological Drugs Overview

Sep 4, 2025

Overview

This lecture covers essential neurological drugs for nursing exams, focusing on mechanisms, key side effects, safe administration, and critical teaching points for patient care.

Anticonvulsants: Phenytoin (Dilantin)

  • Used for long-term seizure prevention (e.g., epilepsy); therapeutic range is 10–20 mcg/mL.
  • Levels <10 risk seizures; >20 risk toxicity—both require HCP notification.
  • Routine blood level and liver function monitoring are required.
  • Early toxicity signs: ataxia (unsteady gait), hand tremor, slurred speech.
  • Adverse effects needing immediate reporting: suicidal thoughts, new/painful rash (Stevens-Johnson syndrome).
  • Normal side effects: gingival hyperplasia (overgrown gums)—teach oral care, use soft toothbrush, inform dentist.
  • Decreases effectiveness of oral contraceptives—use alternative birth control.
  • Do not stop abruptly; taper off to avoid withdrawal seizures.
  • Take at the same time daily; do not administer with tube feedings (hold feeds 1–2 hours before/after, flush with 30–50 mL tap water).
  • Flush IV lines with normal saline pre- and post-administration.
  • Not associated with metallic taste, facial bleeding, or photosensitivity.

Anticonvulsants: Levetiracetam

  • Used for seizure prevention (esp. post-brain tumor/surgery/trauma).
  • Fewer drug interactions than phenytoin.
  • Common side effects: drowsiness, fatigue; avoid driving initially.
  • Report: new anxiety, mood changes, depression, rash/blistering (Stevens-Johnson syndrome).

Cholinesterase Inhibitors: Neostigmine, Pyridostigmine (for Myasthenia Gravis)

  • Increase secretions to improve muscle strength and mobility.
  • Excess can cause cholinergic crisis: salivation, sweating, diarrhea, urinary incontinence, miosis.
  • Antidote for crisis: atropine (anticholinergic).
  • Contraindicated in asthma due to increased secretions/bronchoconstriction.
  • Effectiveness: improved vision and reduced cramping.

Migraine Medications: Sumatriptan, Ergotamine

  • Cause cerebral vasoconstriction to relieve migraines.
  • Contraindicated in CAD and uncontrolled HTN (risk of stroke, MI).
  • Report angina or pale extremities immediately.

Parkinson's Medications: Carbidopa/Levodopa

  • Levodopa increases dopamine; carbidopa prevents its breakdown.
  • Adverse effects: hallucinations, orthostatic hypotension (teach slow position changes).
  • Toxicity: dyskinesia (involuntary movements)—report immediately.
  • Takes 2–6 weeks to take effect; do not stop abruptly.
  • Normal: red/brown urine, sweat, or saliva.
  • Avoid high-protein meals (interferes with absorption).
  • Effectiveness: improved movement/ambulation, not memory.

Anticholinergics: Benztropine, Atropine

  • Reduce secretions and treat tremors in Parkinson’s and extrapyramidal symptoms.
  • Side effects: dry mouth, blurred vision, urinary retention, constipation—“can’t see, can’t pee, can’t spit, can’t poop.”
  • Contraindicated in glaucoma, BPH, and urinary retention.
  • Teach: hydrate, avoid overheating, report urinary retention, rise slowly.

Osmotic Diuretic: Mannitol

  • Lowers intracranial and intraocular pressure.
  • Monitor for heart failure (edema, crackles, pulmonary edema).
  • Give IV only; monitor LOC every hour.

Neuromuscular Blockers: Succinylcholine

  • Used for intubation/paralysis (mechanical ventilation).
  • Does not cause sedation; always sedate with benzodiazepine before use.
  • Life-threatening adverse effect: malignant hyperthermia (muscle rigidity, high fever).
  • Interventions: notify HCP, prepare dantrolene, begin cooling, give oxygen.
  • Screen for personal/family anesthesia reactions and alcoholism prior to use.

Key Terms & Definitions

  • Therapeutic range — safe and effective drug blood level window.
  • Ataxia — unsteady gait or movement.
  • Gingival hyperplasia — gum overgrowth.
  • Cholinergic crisis — excessive secretions due to too much cholinergic medication.
  • Stevens-Johnson syndrome — severe skin reaction with rash/blistering.
  • Dyskinesia — involuntary muscle movements.
  • Malignant hyperthermia — muscle rigidity and high temperature post-anesthesia.
  • Osmotic diuretic — medication removing excess fluid by drawing it into blood vessels.

Action Items / Next Steps

  • Review key drug mechanisms, adverse effects, contraindications, and patient teaching for each class.
  • Commit all critical lab values, side effects, and high-yield tips to memory.
  • Complete assigned readings or practice questions on neurological drugs.
  • Prepare for next lecture/topic as directed by instructor.